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Cat. No. Product Name Target Signaling Pathways
T13156 TG 100572

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100572 is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 nM for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src, Yes, respectively).
T13156L TG 100572 Hydrochloride

VEGFR; FGFR; PDGFR; Src Angiogenesis; Tyrosine Kinase/Adaptors
TG 100572 Hydrochloride 是一种多靶点激酶抑制剂,能够抑制受体酪氨酸激酶和Src 激酶。
T13157 TG 100801

TG100801,TG 100572

VEGFR; Src Angiogenesis; Tyrosine Kinase/Adaptors
TG 100801 是 VEGFr2 和 Src 家族(Src 和 YES)激酶的双重抑制剂,是治疗年龄相关性黄斑变性(AMD)的候选化合物。
T13157L TG 100801 Hydrochloride

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100801 Hydrochloride is a prodrug to treat age-related macular degeneration. TG 100572 is a inhibitor of multi-targeted kinase(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src,

化合物

TG 100572
Cat.No: T13156
Synonym:
Target: VEGFR
TG 100572 Hydrochloride
Cat.No: T13156L
Synonym:
Target: VEGFR, FGFR, PDGFR, Src
TG 100801
Cat.No: T13157
Synonym: TG100801,TG 100572
Target: VEGFR, Src
TG 100801 Hydrochloride
Cat.No: T13157L
Synonym:
Target: VEGFR
TargetMol Loading
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